Mindeudesivir API Manufacturer in India

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Mindeudesivir API

Mindeudesivir, also known as VV116, VV-116, JT001 and deuremidevir, is a deuterated nucleoside analogue antiviral. It was developed as an orally active antiviral compound and is associated with antiviral activity against SARS-CoV-2. Mindeudesivir is the INN name recognized for the compound.

Mindeudesivir is structurally related to remdesivir and contains a deuterium atom in its heterocyclic nucleoside analogue structure. The compound has been investigated and developed particularly for oral antiviral treatment.

Mindeudesivir API Manufacturer in India

Mindeudesivir is a specialized antiviral pharmaceutical API relevant to COVID-19 antiviral research, nucleoside analogue development and pharmaceutical formulation.

Chemical Information

CAS Number: 2647442-33-7
Molecular Formula: C24H30DN5O7
Molecular Weight: 502.54 g/mol
Synonyms: VV116, VV-116, JT001, Deuremidevir
INN: Mindeudesivir
Drug Class: Nucleoside Analogue Antiviral
Therapeutic Area: Antiviral / Infectious Disease
Molecule Type: Deuterated Small Molecule

PubChem lists the compound as C24H31N5O7 because its isotopic notation is represented differently in the database, while the deuterated molecular representation gives C24H30DN5O7 and a molecular weight of approximately 502.5 g/mol.

Mechanism of Action

Mindeudesivir is a nucleoside analogue antiviral. Its molecular design is based on a modified nucleoside analogue that can interfere with viral RNA-dependent replication processes.

Its antiviral research has focused particularly on:

  • SARS-CoV-2
  • Viral RNA replication
  • Nucleoside analogue pharmacology
  • Oral antiviral therapy
  • Coronavirus antiviral development

Pharmaceutical Applications

Mindeudesivir has been associated with pharmaceutical research and development involving:

  • COVID-19
  • SARS-CoV-2 infection
  • Antiviral drug development
  • Coronavirus research
  • Nucleoside analogue therapeutics
  • Oral antiviral formulations

Mindeudesivir/deuremidevir has received regulatory recognition in China, with IUPHAR listing it as an approved drug in China in 2023.

Dosage Form Applications

Mindeudesivir has been developed for oral administration, including formulations containing its hydrobromide salt.

Physical Characteristics

Mindeudesivir free base is described as a solid, with a reported molecular weight of approximately 502.54 g/mol for the deuterated form. Commercial research documentation describes the material as white to off-white.

Manufacturing Process

A controlled Mindeudesivir API manufacturing process may involve:

  1. Qualification of starting materials
  2. Preparation of protected nucleoside intermediates
  3. Controlled incorporation of the deuterium isotope
  4. Glycosylation / nucleoside analogue construction
  5. Introduction of the nitrile functionality
  6. Esterification
  7. Deprotection
  8. Purification
  9. Salt formation where applicable
  10. Crystallization
  11. Controlled drying
  12. Final analytical characterization
  13. Pharmaceutical-grade packaging

Quality Control Testing

For Mindeudesivir API, analytical characterization may include:

  • Identification by IR
  • HPLC identification
  • LC-MS
  • Assay
  • Related substances
  • Deuterium-isotope incorporation / isotopic purity
  • Water content
  • Residual solvents
  • Elemental impurities
  • Specific optical rotation
  • Chiral purity
  • Stability testing

Storage

Store Mindeudesivir under controlled pharmaceutical storage conditions, protected from moisture, excessive heat and direct light. Exact storage conditions should be established from validated stability data for the specific API form.

Pharmaceutical Research

Mindeudesivir is relevant to:

  • SARS-CoV-2 antiviral research
  • Coronavirus drug development
  • Nucleoside analogue pharmacology
  • RNA-dependent RNA polymerase research
  • Deuterated drug development
  • Oral antiviral formulation
  • Infectious-disease pharmaceutical research

Detailed Specifications

Parameter Specification
Appearance White crystalline powder or crystals
Identification IR & HPLC compliant
Assay (HPLC) 99.0–100.5%
Loss on Drying NMT 1.0%
Residue on Ignition NMT 0.1%
pH (1% Solution) 3.2–3.5
Specific Rotation +31.5° to +33.5° at 405 nm
Melting Point 171–175°C
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