Estrone-3-Sulphate API Manufacturer & Supplier in India

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Estrone-3-Sulphate API Manufacturer & Supplier in India

Estrone-3-Sulphate is a sulfate conjugate of estrone, an endogenous steroidal estrogen. It is an estrogen metabolite and serves as an important intermediate and reservoir form of estrogen in biological systems. Estrone-3-sulfate is also used in pharmaceutical and biochemical research applications.

Estrone-3-sulfate can undergo enzymatic conversion to estrone, which may subsequently participate in estrogenic signaling. Its sulfate-conjugated structure influences its solubility, transport and metabolism.

What is Estrone-3-Sulphate?

Estrone-3-Sulphate is the 3-sulfate ester of estrone. It belongs to the family of steroid sulfate conjugates and is formed naturally through sulfation of estrone.

CAS Number: 481-97-8
Molecular Formula: C₁₈H₂₂O₆S
Molecular Weight: 366.43 g/mol

Mechanism / Biological Activity

Estrone-3-sulfate itself is a conjugated, relatively inactive estrogen reservoir. It can be hydrolyzed by steroid sulfatase (STS) to generate estrone, which can then contribute to estrogen receptor-mediated activity.

Its biological relevance includes:

  • Conversion to estrone through steroid sulfatase
  • Participation in estrogen metabolism
  • Serving as a circulating estrogen reservoir
  • Contribution to local estrogen availability
  • Indirect involvement in estrogen receptor signaling

Pharmaceutical & Research Applications

Estrone-3-Sulphate may be used in:

  • Steroid hormone research
  • Estrogen metabolism studies
  • Pharmaceutical research
  • Biochemical and analytical research
  • Development and evaluation of estrogen-related compounds
  • Reference and analytical applications

Its exact use depends on the grade, specification and intended application.

Estrone-3-Sulphate API / Pharmaceutical Raw Material

Estrone-3-Sulphate is a steroidal sulfate conjugate with defined chemical structure and stereochemistry. Quality evaluation should control identity, purity, related substances, water content and other applicable quality attributes.

Typical analytical evaluation may include:

  • Identification
  • Assay
  • Related substances
  • Water content
  • Residual solvents
  • Specific optical rotation, where applicable
  • Sulfate content, where applicable
  • Elemental impurities
  • Particle-size characteristics, where applicable

Quality & Regulatory Considerations

Pharmaceutical or research-grade Estrone-3-Sulphate should comply with the applicable approved specification and intended-use requirements.

A qualified supplier should provide Certificate of Analysis (CoA), specification sheet, SDS/MSDS, batch traceability and applicable regulatory documentation.

Storage

Store Estrone-3-Sulphate in a tightly closed container, protected from moisture, excessive heat and direct light, according to the applicable manufacturer-approved storage conditions.

Detailed Specifications

Parameter Specification
Appearance White to off-white crystalline powder
Identification IR & HPLC compliant
Assay (HPLC) 98.0% – 102.0%
Loss on Drying NMT 1.0%
Residue on Ignition NMT 0.5%
Heavy Metals NMT 20 ppm
pH (1% Solution) 2.0 – 4.0
Total Impurities NMT 1.0%
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